Raltegravir

In the US, Raltegravir (raltegravir systemic) is a member of the drug class integrase strand transfer inhibitor and is used to treat HIV Infection.

US matches:

• Raltegravir


• Raltegravir Potassium

Scheme

Rec.INN

ATC (Anatomical Therapeutic Chemical Classification)

J05AX08

CAS registry number (Chemical Abstracts Service)

0518048-05-0

Chemical Formula

C20-H21-F-N6-O5

Molecular Weight

444

Therapeutic Category

Antiviral agent, treatment of HIV infection

Chemical Names

N-[(4-Fluorophenyl)methyl]-5-hydroxy-1-methyl-2-[2-(5-methyl-1,3,4-oxadiazole-2-carboxamido)propan-2-yl]-6-oxo-1,6-dihydropyrimidine-4-carboxamide (WHO)

4-Pyrimidinecarboxamide, N-((4-fluorophenyl)methyl)-1,6-dihydro-5-hydroxy-1-methyl-2-(1-methyl-1-(((5-methyl-1,3,4-oxadiazol-2-yl)carbonyl)amino)ethyl)-6-oxo-

5-Hydroxy-1-methyl-2-{1-methyl-1-[(5-methyl[1,3,4]oxadiazol-2-carbonyl)amino]ethyl}-6-oxo-1,6-dihydropyrimidin-4-carbonsäure-4-fluorbenzylamid (IUPAC)

N-(2-(4-(4-Fluorobenzylcarbamoyl)-5-hydroxy-1-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)propan-2-yl)-5-methyl-1,3,4-oxadiazole-2-carboxamide

Foreign Names

• Raltegravirum (Latin)
• Raltegravir (German)
• Raltégravir (French)
• Raltegravir (Spanish)

Generic Names

• Raltegravir (OS: BAN)
• c-1605 (IS)
• MK-0518 (IS)
• MK-518 (IS: Merck)
• Raltegravir Potassium (OS: USAN)
• 4-Pyrimidinecarboxamide (IS)

Brand Names

• Isentress
  Merck, United States; Merck Sharp & Dohme, Belgium; Merck Sharp & Dohme, Greece; Merck Sharp & Dohme, Netherlands; Merck Sharp & Dohme, Slovenia; MSD, Denmark; Merck Frosst, Canada; Merck Sharp & Dohme, Austria; Merck Sharp & Dohme, Australia; Merck Sharp & Dohme, Germany; Merck Sharp & Dohme, France; Merck Sharp & Dohme, United Kingdom; Merck Sharp & Dohme, Croatia (Hrvatska); Merck Sharp & Dohme, Ireland; Merck Sharp & Dohme, Italy; Merck Sharp & Dohme, Peru; Merck Sharp & Dohme, Sweden; MSD, Switzerland; MSD, Norway

International Drug Name Search

Glossary

BAN	British Approved Name
IUPAC	International Union of Pure and Applied Chemistry
IS	Inofficial Synonym
OS	Official Synonym
Rec.INN	Recommended International Nonproprietary Name (World Health Organization)
USAN	United States Adopted Name
WHO	World Health Organization

Click for further information on drug naming conventions and International Nonproprietary Names.